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No longer recruiting (closed or complete)Last updated: 8 August 2025

FPI-2265-203: A study investigating how safe, effective and tolerable a drug that delivers targeted radiation to cancer cells (called FPI-2265) is when given in combination with another targeted therapy (called Olaparib) in people with metastatic castration-resistant prostate cancerA Phase 2, Open-label, Multi-centre Study of FPI-2265 (225Ac-PSMA-I&T) and Olaparib in Participants With Metastatic Castration Resistant Prostate Cancer (mCRPC)

Trial purpose

Medical clipboardCancer treatment

Tumor type

Urinary System Cancers Genitourinary

Age

People18+

Trial acronym

FPI-2265-203

Clinical summary

Summary

This study will be conducted in two parts, and each part will be evaluating two treatment regimens.

The part of the study you are assigned to is based on whether or not you have previously had treatment with lutetium-177 (177Lu) vipivotide tetraxetan or other 177Lu-PSMA radioligand therapy (RLT). Those who have had prior treatment with these agents will enrol in Part A, and those who have not will enrol in Part B.

For each part of the study, a Simon 2-stage design will be used to evaluate two dosing regimens. Participants with PSMA-positive metastatic castration-resistant prostate cancer (mCRPC) will be allocated to Arm 1 and Arm 2 in a singular, alternating fashion, until all Stage 1 participants are enrolled into each of the two regimens:

  • Arm 1: Will consist of up to 6 doses of FPI-2265 every 6 weeks at Dose A and Olaparib twice a day on Days 1 and 14 of each cycle.
  • Arm 2: Will consist of up to 9 doses of FPI-2265 every 4 weeks at Dose B and Olaparib twice a day on Days 1 and 14 of each cycle.

Participants will be monitored and assessed for efficacy response, disease progression and adverse events.

Conditions

This trial is treating people with metastatic castration-resistant prostate cancer

Eligibility

Inclusion

  1. Adult male participants with mCRPC that is progressing at the time of study entry
  2. ECOG performance status 0-1 and life expectancy of at least three months
  3. Must have received at least one novel anti-androgen deprivation therapy
  4. Participants with known BRCA mutations should have received approved therapies such as PARP inhibitors, per Investigator discretion.
  5. All prior treatment-related AEs must have resolved to CTCAE Grade ≤1 (except alopecia).
  6. Participants must have had prior orchiectomy and/or ongoing androgen deprivation therapy and a castrate level of serum testosterone (<50 ng/dL or <1.7 nmol/L)
  7. Positive PSMA PET/CT scans .
  8. Participants must have adequate organ and bone marrow function:

    • Hgb >/= 9g/dL
    • Platelets >/= 100 x 10^9/L
    • ANC </= 1.5 x 10^9/L
    • CrCL >/= 50 mL/min

Exclusion

  1. Previous treatment with any of the following within 6 months of first dose: Samarium-153, Rhenium-186, Rhenium-188, Radium-223, hemi-body irradiation.
  2. Participants who received more than two (2) prior lines of cytotoxic chemotherapy for CRPC.
  3. Participants with known unresolved urinary tract obstruction.
  4. Transfusion- or growth factor-dependent participants.
  5. Participants with a history of CNS metastases are excluded, except those who have received therapy (and are neurologically stable, asymptomatic, and not receiving corticosteroids for the purposes of maintaining neurologic integrity.
  6. Symptomatic cord compression, or clinical or radiologic findings indicative of impending cord compression.
  7. Participants with any liver metastases.
  8. Participants with skeletal metastases presenting as a superscan .
  9. Previous history of interstitial lung disease or non-infectious pneumonitis.
  10. Participants with a history or clinical and/or laboratory features suggestive of MDS/AML.
  11. Major surgery ≤28 days prior to the first dose of study treatment.
  12. Planning to conceive a pregnancy during the treatment and up to six months after the last treatment.
  13. Participants unable to swallow orally administered medications or with malabsorptive gastrointestinal disorders.
  14. Concomitant use of known strong or moderate CYP3A inhibitors or inducers

Inclusion

  • Your cancer has spread to other parts of the body (metastatic) or has grown into nearby parts of the body (locally advanced).
  • You have had treatment but your cancer has gotten worse or has not responded to the treatment you have been given.
  • You have had a certain type of treatment or surgical procedure.

Exclusion

  • You have certain types of non-cancer medical conditions.
  • You have had certain treatments, surgical procedures or drugs.
Message

Clinical trials have complex eligibility criteria, and other criteria may apply for this trial. Ask your doctor about whether this trial could be right for you.

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More information

Trial Identifiers

Information on this page is partially produced from ClinicalTrials.gov *. View further details about this trial on the registry via the links below:

Trial sponsor

Fusion Pharmaceuticals Inc.

Scientific Title

A Phase 2, Open-label, Multi-centre Study of FPI-2265 (225Ac-PSMA-I&T) and Olaparib in Participants With Metastatic Castration Resistant Prostate Cancer (mCRPC)

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